LKT Labs

Biochemicals for Life Science Research

MLN2480

MLN2480

Product ID M4452
Cas No. 1096708-71-2
Purity ≥98%
Product Unit SizeCostQuantityStock
1 mg $90.00 In stock
5 mg $299.60 In stock
Bulk Quote

Quicklinks

Description

MLN2480 is an oral pan-Raf inhibitor designed to inhibit cell proliferation and survival. MLN2480 is currently in clinical trials and displays anticancer chemotherapeutic activity.

Product Info

Cas No.

1096708-71-2
Purity

≥98%
Formula

C17H12Cl2F3N7O2S
Formula Wt.

506.30
IUPAC Name

2-[(1R)-1-[(6-amino-5-chloropyrimidine-4-carbonyl)amino]ethyl]-N-[5- chloro-4-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole-5-carboxamide
Solubility

DMSO 100 mg/mL (197.51 mM) Ethanol 100 mg/mL (197.51 mM) Water Insoluble

Shipping and Storage

Store Temp

-20°C
Ship Temp

Ambient

Downloads

MSDS

M4452 MSDS PDF
Info Sheet

M4452 Info Sheet PDF
Brochures

Ras-Raf-MEK-ERK Pathway Booklet

References

http://clinicaltrials.gov/show/NCT01425008

Custom Order

  • Size of single unit expressed as number (e.g. '500' in the case of 500 mg)
  • Total quantity of unit size desired (e.g. '10' in the case of 10 x 500 mg). If only one unit is desired, you may leave this blank.
  • This field is for validation purposes and should be left unchanged.

Related Products

  • D4873

    Meso-2,3-dimercaptosuccinic Acid

    Organosulfur, chelating agent.
    ≥98%
  • C2949

    Chlorpheniramine Maleate

    Alkylamine; histamine H1 antagonist, SERT and NET ...
    ≥98%
  • N0212

    Nedaplatin

    Pt-based DNA cross-linker.
    ≥98%
  • A4400

    Alamethicin

    Antimicrobial peptide found in Trichoderma, induce...
    ≥95%
  • L5660

    Loperamide Hydrochloride

    FIASMA, μOR agonist, potential HCN channel blocke...
    ≥98%
  • A5373

    Anisomycin

    Peptidyl transferase inhibitor, protein translatio...
    ≥98%
  • T1020

    n-Butyl Analog of Paclitaxel

    n-Butyl Analog of Paclitaxel is an impurity of the...
    ≥95%
  • N1985

    Neuropeptide K, pig

    Endogenous peptide, N-terminal-extended neurokinin...
    ≥95%
  • A5287

    Angiotensinogen (1-14), human

    Peptide fragment, renin substrate, precursor to AT...
    ≥95%
  • J889280

    JWH 015

    Cannabinoid receptor 2 selective agonist.
    ≥98%
  • A5458

    Anorexigenic Peptide

    Peptide, alters hormone secretion and feeding beha...
    ≥95%
  • C0372

    Casein Kinase 2 Assay Kit

    Casein kinase 2 substrate.
    ≥95%
  • P0397

    Pazopanib

    VEGFR, PDGFR, c-Kit inhibitor.
    ≥97%
  • A7072

    Atriopeptin III

    ANP analog, cardiomodulatory peptide; NPR-A agonis...
    ≥95%
  • A0249

    BAM-22P

    Peptide, cleavage product of proenkephalin; κOR a...
    ≥95%
  • G0106

    Gabapentin

    GABA analog; GABA potentiator, adenosine A1 agonis...
    ≥98%
  • R0250

    Ranatensin

    Peptide found in amphibians.
    ≥98%
  • M1687

    Mevinolin

    Statin, naturally produced by mushrooms; HMG-CoA r...
    ≥97%
  • B6807

    [Des-Arg9]-Bradykinin

    Natriuretic, vasodilatory peptide, bradykinin anal...
    ≥95%
  • C1869

    Cerulenin

    Found in Cephalosporium; fatty acid synthase inhib...
    ≥98%